An adenylyl cyclase 1 (AC1) and AC6 inhibitor; selective for AC1 and AC6

CB-7921220 – 1 mg

Brand:
Cayman
CAS:
115453-99-1
Storage:
-20
UN-No:
Non-Hazardous - /

CB-7921220 is an inhibitor of the adenylyl cyclase (AC) isoforms AC1 and AC6.{38294} It is selective, reducing AC1 and AC6 activity by 60% while having no effect on AC2 and AC5 in Sf9 membranes stimulated by forskolin (Item No. 11018) when used at a concentration of 100 μM.  

 

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SKU: 23332 - 1 mg Category:

Description

An adenylyl cyclase 1 (AC1) and AC6 inhibitor; selective for AC1 and AC6, reducing their activity by 60% while having no effect on AC2 and AC5 in Sf9 membranes stimulated by forskolin (Item No. 11018) at 100 µM, ,

Formal name: 6-[2-(4-aminophenyl)ethenyl]-2-pyridinecarboxylic acid

Synonyms: 

Molecular weight: 240.3

CAS: 115453-99-1

Purity: ≥98%

Formulation: A crystalline solid

Product Type|Biochemicals|Small Molecule Inhibitors|Nucleic Acid Turnover/Signaling||Research Area|Cell Biology|Cell Signaling|cAMP Signaling

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