An LPA mimetic

Oleoyl Ethanolamide Phosphate – 5 mg

Brand:
Cayman
CAS:
24435-25-4
Storage:
-20
UN-No:
Non-Hazardous - /

Oleoyl ethanolamide phosphate (OEA-P) is a lysophosphatidic acid (LPA) mimetic, LPA receptor agonist, and phosphate ester of oleoyl ethanolamide (OEA; Item No. 90265).{47608,7616} It selectively increases [35S]GTPγS binding to HEK293T cell membranes expressing LPA1 and LPA2 over LPA3 receptors.{7616} OEA-P induces calcium mobilization and inhibits forskolin-induced cAMP accumulation in MDA-MB-231 cells (EC50s = 1.2 and 101 nM, respectively).{47608}  

 

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SKU: 22886 - 5 mg Category:

Description

An LPA mimetic, LPA receptor agonist, and phosphate ester of OEA; selectively increases [35S]GTPγS binding to HEK293T cell membranes expressing LPA1 and LPA2 over LPA3 receptors; induces calcium mobilization and inhibits forskolin-induced cAMP accumulation in MDA-MB-231 cells (EC50s = 1.2 and 101 nM, respectively)

Formal name: N-[2-(phosphonooxy)ethyl]-9Z-octadecenamide

Synonyms:  NAEPA|N-oleoyl ethanolamide phosphoric acid|OEA-P

Molecular weight: 405.5

CAS: 24435-25-4

Purity: ≥95%

Formulation: A crystalline solid

Product Type|Biochemicals|Lipids|Fatty Amides||Product Type|Biochemicals|Receptor Pharmacology|Agonists||Research Area|Lipid Biochemistry|Endocannabinoid/Endocannabinoid-like||Research Area|Lipid Biochemistry|Glycerophospholipids

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