An amphetamine that acts as an agonist at serotonin (5-HT) receptors (IC50s = 6.92

3-Trifluoromethylamphetamine (hydrochloride) – 1 mg

Brand:
Cayman
CAS:
673-18-7
Storage:
-20
UN-No:
Non-Hazardous - /

3-Trifluoromethylamphetamine (hydrochloride) ( Item No. 22604) is an analytical reference standard that is categorized as an amphetamine. It is an active metabolite of fenfluramine and benfluorex that acts as an agonist at serotonin (5-HT) receptors (IC50s = 6.92, 3.55, 0.17, and 2.09 µM for 5-HT1A, 5-HT1B, 5-HT1C, and 5-HT2 receptors, respectively, in murine brain).{39006,39005} Norfenfluramine induces anorexia in mice and rats with EC50 values of 6.8 and 0.8 mg/kg, i.p., respectively.{39006} This product is intended for research and forensic applications.  

 

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Description

An amphetamine that acts as an agonist at serotonin (5-HT) receptors (IC50s = 6.92, 3.55, 0.17, and 2.09 µM for 5-HT1A, 5-HT1B, 5-HT1C, and 5-HT2 receptors, respectively, in murine brain); induces hypophagia in mice and rats with EC50 values of 6.8 and 0.8 mg/kg, i.p., respectively,

Formal name: α-methyl-3-(trifluoromethyl)-benzeneethanamine, monohydrochloride

Synonyms:  (±)-Norfenfluramine|desethyl Fenfluramine

Molecular weight: 239.7

CAS: 673-18-7

Purity: ≥98%

Formulation: A crystalline solid

Application|Mass Spectrometry||Product Type|Biochemicals|Analytical Standards||Product Type|Biochemicals|Drugs of Abuse||Research Area|Forensic Chemistry & Toxicology|Performance-Enhancing Drugs|Stimulants||Research Area|Forensic Chemistry & Toxicology|Stimulants|Amphetamines

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