An internal standard for the quatification of tolperisone by GC- or LC-MS

Tolperisone-d10 (hydrochloride) – 1 mg

Brand:
Cayman
CAS:
1185160-65-9
Storage:
2-8
UN-No:
Non-Hazardous - /

Tolperisone-d10 is intended for use as an internal standard for the quantification of tolperisone by GC- or LC-MS. Tolperisone is a piperidine that acts as an inhibitor of voltage-gated sodium channels with an IC50 value of 198 µM, for inhibition of peak sodium currents evoked by step depolarizations in dorsal root ganglion (DRG) neurons, in vitro.{34788} Tolperisone acts as an antispastic agent that attenuates monosynaptic, disynaptic, and polysynaptic reflux response to dorsal root stimulation in vivo. Formulations containing tolperisone are used as analgesics and muscle relaxants.  

 

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Description

An internal standard for the quatification of tolperisone by GC- or LC-MS

Formal name: 3-2,2,3,3,4,4,5,5,6,6-decadeuteriopiperidin-1-yl)-2-methyl-1-(4-methylphenyl)propan-1-one, monohydrochloride)

Synonyms: 

Molecular weight: 291.9

CAS: 1185160-65-9

Purity: ≥99% deuterated forms (d1-d10)

Formulation: A solid

Application|Mass Spectrometry||Product Type|Biochemicals|Ion Channel Modulation|Blockers||Product Type|Biochemicals|Isotopically Labeled Standards|Deuterium||Research Area|Neuroscience|Pain Research

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