A potent inhibitor of recombinant FGFR4 (IC50 50 < 10 nM)

BLU-554 – 10 mg

Brand:
Cayman
CAS:
1707289-21-1
Storage:
-20
UN-No:
Non-Hazardous - /

BLU-554 is a potent inhibitor of recombinant fibroblast growth factor receptor 4 (FGFR4; IC50 50 < 10 nM), a marker of FGFR4 inhibition, in MDA-MB-453 breast cancer cells.  

 

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SKU: 22438 - Category:

Description

A potent inhibitor of recombinant FGFR4 (IC50 50 < 10 nM), a marker of FGFR4 inhibition, in MDA-MB453 cells,

Formal name: N-[(3S,4S)-3-[[6-(2,6-dichloro-3,5-dimethoxyphenyl)-2-quinazolinyl]amino]tetrahydro-2H-pyran-4-yl]-2-propenamide

Synonyms: 

Molecular weight: 503.4

CAS: 1707289-21-1

Purity: ≥95%

Formulation: A crystalline solid

Product Type|Biochemicals|Kinase Inhibitors|FGFR Family||Product Type|Biochemicals|Small Molecule Inhibitors|Kinases||Research Area|Cancer|Cell Signaling|Growth Factor Receptor Signaling

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