An isomer of fluoxetine; has weaker SSRI activity than fluoxetine (Kis = 166 and 17 nM

meta-Fluoxetine (hydrochloride) – 10 mg

Brand:
Cayman
CAS:
79088-29-2
Storage:
-20
UN-No:
Non-Hazardous - /

meta-Fluoxetine is an isomer of fluoxetine (Item No. 14418) that is found as an impurity in fluoxetine preparations. meta-Fluoxetine is a weaker serotonin selective reuptake inhibitor (SSRI) than fluoxetine, in which the trifluoromethyl group is at the para position (Kis = 166 and 17 nM, respectively, in rat brain synaptosomes).{36026,36027}  

 

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Description

An isomer of fluoxetine; has weaker SSRI activity than fluoxetine (Kis = 166 and 17 nM, respectively, in rat brain synaptosomes)

Formal name: N-methyl-γ-[3-(trifluoromethyl)phenoxy]-benzenepropanamine, monohydrochloride

Synonyms:  m-Fluoxetine|Fluoxetine Impurity C|Fluoxetine Related Compound A

Molecular weight: 345.8

CAS: 79088-29-2

Purity: ≥98%

Formulation: A crystalline solid

Product Type|Biochemicals|Transporter & Exchanger Modulators||Research Area|Neuroscience|Behavioral Neuroscience|Anxiety||Research Area|Neuroscience|Behavioral Neuroscience|Depression

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