A Ca2+ channel activator; a racemic mixture of the (R)-(+)-BAY-K-8644 and (S)-(−)-BAY-K-8644 versions; has similar effects as (S)-(−)-BAY-K-8644; demonstrates vasoconstrictive and positive inotropic effects in vivo; has behavioral effects

(±)-BAY-K-8644 – 5 mg

Brand:
Cayman
CAS:
71145-03-4
Storage:
-20
UN-No:
Non-Hazardous - /

(±)-BAY-K-8644 is a racemic mixture composed of two optical isomers, (R)-(+)-BAY-K-8644 (Item No. 15263) and (S)-(−)-BAY-K-8644 (Item No. 19988). (±)-BAY-K-8644 has similar effects as (S)-(−)-BAY-K-8644, which activates voltage-sensitive L-type calcium channels.{37139,37140} (±)-BAY-K-8644 and (S)-(−)-BAY-K-8644 also demonstrate vasoconstrictive and positive inotropic effects in vivo as well as behavioral effects, including deficits to motor function.{24673,24674}  

 

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Description

A Ca2+ channel activator; a racemic mixture of the (R)-(+)-BAY-K-8644 and (S)-(−)-BAY-K-8644 versions; has similar effects as (S)-(−)-BAY-K-8644; demonstrates vasoconstrictive and positive inotropic effects in vivo; has behavioral effects, including deficits to motor function

Formal name: 1,4-dihydro-2,6-dimethyl-5-nitro-4-[2-(trifluoromethyl)phenyl]-3-pyridinecarboxylic acid, methyl ester

Synonyms:  SQ 28,873

Molecular weight: 356.3

CAS: 71145-03-4

Purity: ≥98%

Formulation: A crystalline solid

Product Type|Biochemicals|Ion Channel Modulation|Activators||Research Area|Cardiovascular System|Heart|Myocardial Contractility||Research Area|Cardiovascular System|Vasculature|Vasoconstriction||Research Area|Neuroscience|Behavioral Neuroscience

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