A potent

CNX-774 – 1 mg

Brand:
Cayman
CAS:
1202759-32-7
Storage:
-20
UN-No:
Non-Hazardous - /

CNX-774 is a potent, selective, and irreversible inhibitor of Bruton’s tyrosine kinase (BTK), an important kinase in the B cell antigen receptor pathway, with IC50 values of 50 = 2.82 and 0.38 µM) but has no effect on cell cycle progression.{34333}  

 

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Description

A potent, selective, and irreversible BTK inhibitor

Formal name: 4-[4-[[5-fluoro-4-[[3-[(1-oxo-2-propen-1-yl)amino]phenyl]amino]-2-pyrimidinyl]amino]phenoxy]-N-methyl-2-pyridinecarboxamide

Synonyms: 

Molecular weight: 499.5

CAS: 1202759-32-7

Purity: ≥98%

Formulation: A crystalline solid

Product Type|Biochemicals|Kinase Inhibitors|Tec Family||Product Type|Biochemicals|Small Molecule Inhibitors|Kinases||Research Area|Cancer|Cell Signaling|Tec Family Signaling||Research Area|Cell Biology|Cell Signaling

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