An NSAID that inhibits both isoforms of COX (IC50s = 1.1 and 8.7 µM for COX-1 and COX-2

Suprofen – 5 mg

Brand:
Cayman
CAS:
40828-46-4
Storage:
-20
UN-No:
- 2811 / 6.1

Suprofen is a non-steroidal anti-inflammatory drug (NSAID) that non-selectively inhibits both isoforms of cyclooxygenase (COX; IC50s = 1.1 and 8.7 µM for COX-1 and COX-2, respectively).{8427,1286}  

 

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Description

An NSAID that inhibits both isoforms of COX (IC50s = 1.1 and 8.7 µM for COX-1 and COX-2, respectively)

Formal name: α-methyl-4-(2-thienylcarbonyl)-benzeneacetic acid

Synonyms:  (±)-Suprofen|NSC 303611|R 25061|TN 762

Molecular weight: 260.3

CAS: 40828-46-4

Purity: ≥98%

Formulation: A crystalline solid

Product Type|Biochemicals|Small Molecule Inhibitors|Cyclooxygenases||Research Area|Immunology & Inflammation|Inflammatory Lipid Mediators|Prostaglandins||Research Area|Lipid Biochemistry|Cyclooxygenase Pathway

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