A dihydropyridine L-type calcium channel blocker with a slow onset profile that displays antihypertensive activity

Azelnidipine – 1 g

Brand:
Cayman
CAS:
123524-52-7
Storage:
-20
UN-No:
Non-Hazardous - /

Azelnidipine is a third generation, dihydropyridine L-type calcium channel blocker with a slow onset profile that displays long-lasting antihypertensive activity in hypertensive rat models compared to other L-type calcium channel blockers.{33379,33378}  

 

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Description

A dihydropyridine L-type calcium channel blocker with a slow onset profile that displays antihypertensive activity

Formal name: 2-amino-1,4-dihydro-6-methyl-4-(3-nitrophenyl)-3,5-pyridinedicarboxylic acid, 3-[1-(diphenylmethyl)-3-azetidinyl] 5-(1-methylethyl) ester

Synonyms:  CS 905|RS 9054

Molecular weight: 582.7

CAS: 123524-52-7

Purity: ≥98%

Formulation: A crystalline solid

Product Type|Biochemicals|Ion Channel Modulation|Blockers||Research Area|Cardiovascular System|Cardiovascular Diseases|Hypertension

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