A histamine receptor antagonist (Ki = 142 nM for H4) and calcium channel blocker that potently dilates peripheral vessels

Cinnarizine – 25 g

Brand:
Cayman
CAS:
298-57-7
Storage:
22
UN-No:
Non-Hazardous - /

Cinnarizine is a piperazine derivative that has diverse cellular and physiological actions. It is a histamine (H) receptor antagonist (Ki = 142 nM for H4) and calcium channel blocker that potently dilates peripheral vessels.{22485,30252,32995} Formulations containing cinnarizine have been used to manage vertigo, nausea, and migraines.{30252,32996}  

 

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SKU: 21001 - Category:

Description

A histamine receptor antagonist (Ki = 142 nM for H4) and calcium channel blocker that potently dilates peripheral vessels

Formal name: 1-(diphenylmethyl)-4-(3-phenyl-2-propen-1-yl)-piperazine

Synonyms: 

Molecular weight: 368.5

CAS: 298-57-7

Purity: ≥98%

Formulation: A crystalline solid

Product Type|Biochemicals|Ion Channel Modulation|Blockers||Product Type|Biochemicals|Receptor Pharmacology|Antagonists||Research Area|Cardiovascular System|Cardiovascular Diseases||Research Area|Cardiovascular System|Vasculature|Vasoconstriction||Research Area|Cardiovascular System|Vasculature|Vasodilation||Research Area|Cell Biology|Cell Signaling|Calcium Mobilization||Research Area|Neuroscience|Pain Research

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