An alkaloid that has been described as an inhibitor of phosphodiesterase 4 and negative allosteric modulator of L-type Ca2+ channels; used as an antispasmodic to help cervical dilation in the early stages of labor

Drotaverine (hydrochloride) – 500 mg

Brand:
Cayman
CAS:
985-12-6
Storage:
-20
UN-No:
Non-Hazardous - /

Drotaverine is an alkaloid that has been described as an inhibitor of phosphodiesterase 4 and negative allosteric modulator of L-type Ca2+ channels.{33092,33094} Formulations containing drotaverine are used as antispasmodics to help cervical dilation in the early stages of labor.{33093}  

 

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Description

An alkaloid that has been described as an inhibitor of phosphodiesterase 4 and negative allosteric modulator of L-type Ca2+ channels; used as an antispasmodic to help cervical dilation in the early stages of labor

Formal name: 1-[(3,4-diethoxyphenyl)methylene]-6,7-diethoxy-1,2,3,4-tetrahydro-isoquinoline, monohydrochloride

Synonyms: 

Molecular weight: 434

CAS: 985-12-6

Purity: ≥98%

Formulation: A crystalline solid

Product Type|Biochemicals|Ion Channel Modulation|Blockers||Product Type|Biochemicals|Small Molecule Inhibitors|MMPs||Product Type|Biochemicals|Small Molecule Inhibitors|Phosphodiesterases||Research Area|Endocrinology & Metabolism|Reproductive Biology

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