An antimalarial drug that is used in combination with artemether

Lumefantrine – 1 g

Brand:
Cayman
CAS:
82186-77-4
Storage:
-20
UN-No:
Non-Hazardous - /

Lumefantrine is an antimalarial drug that is used in combination with artemether (Item No. 11815).{26532} The pairing of lumefantrine and artemether is a major form of oral artemisinin combination therapy used against uncomplicated P. falciparum malaria.{28281,21234} Lumefantrine also blocks the rapidly activating delayed-rectifier potassium channel (IKr; IC50 = 8.1 µM).{24505}  

 

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Description

An antimalarial drug that is used in combination with artemether

Formal name: (9Z)-2,7-dichloro-9-[(4-chlorophenyl)methylene]-α-[(dibutylamino)methyl]-9H-fluorene-4-methanol

Synonyms:  Benflumetol|CPG-56695

Molecular weight: 528.9

CAS: 82186-77-4

Purity: ≥98%

Formulation: A crystalline solid

Product Type|Biochemicals|Antiparasitics|Antiprotozoals||Product Type|Biochemicals|Ion Channel Modulation|Blockers||Research Area|Immunology & Inflammation||Research Area|Infectious Disease|Parasitic Diseases|Malaria

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