A stable derivative of apoptolidin (Item No. 19435) that demonstrates 10-fold reduced F1FO-ATP synthase inhibitory activity compared to apoptolidin (IC50s = 17 and 0.7 µM

Isoapoptolidin – 100 µg

Brand:
Cayman
CAS:
476647-30-0
Storage:
-20
UN-No:
Non-Hazardous - /

Isoapoptolidin is a stable derivative of apoptolidin (Item No. 19435) that demonstrates 10-fold reduced F1FO-ATP synthase inhibitory activity compared to apoptolidin (IC50s = 17 and 0.7 µM, respectively).{32128,32129}  

 

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SKU: 20590 - Category:

Description

A stable derivative of apoptolidin (Item No. 19435) that demonstrates 10-fold reduced F1FO-ATP synthase inhibitory activity compared to apoptolidin (IC50s = 17 and 0.7 µM, respectively)

Formal name: (3E,5E,7E,9R,10R,11E,13E,17S,18S,20S,21R)-10-[(6-deoxy-4-O-methyl-α-L-glucopyranosyl)oxy]-21-[O-2,6-dideoxy-3-O-methyl-β-D-arabino-hexopyranosyl-(1→4)-O-2,6-dideoxy-3-C-methyl-α-L-arabino-hexopyranosyl-(1→7)-2,4,6-trideoxy-1-C-hydroxy-2,4-dimethyl-8-O-methyl-L-glycero-β-D-galacto-octopyranosyl]-17,20-dihydroxy-18-methoxy-3,5,7,9,13-pentamethyl-oxacycloheneicosa-3,5,7,11,13-pentaen-2-one

Synonyms: 

Molecular weight: 1,129.40

CAS: 476647-30-0

Purity: ≥90%

Formulation: A lyophilisate

Product Type|Biochemicals|Small Molecule Inhibitors|MMPs||Product Type|Biochemicals|Small Molecule Inhibitors|Oxidative Phosphorylation||Research Area|Cell Biology|Mitochondrial Biology

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