A natural metabolite of dopamine; a weak agonist of TAAR1 (EC50 = 1.7 µM)

3-methoxy Tyramine (hydrochloride) – 50 mg

Brand:
Cayman
CAS:
1477-68-5
Storage:
-20
UN-No:
Non-Hazardous - /

3-methoxy Tyramine is a natural metabolite of dopamine, produced by catechol O-methyltransferase (COMT). It is a weak agonist of trace amine-associated receptor 1 (EC50 = 1.7 µM).{29548} 3-methoxy Tyramine levels are assessed to monitor COMT activity in Parkinson’s disease.{32113} Elevated 3-methoxy Tyramine levels may also indicate abnormal catecholamine synthesis that occurs in certain neuroendocrine tumors.{32114}  

 

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Description

A natural metabolite of dopamine; a weak agonist of TAAR1 (EC50 = 1.7 µM)

Formal name: 4-(2-aminoethyl)-2-methoxy-phenol, monohydrochloride

Synonyms:  3-O-methyl Dopamine|3-Methoxy-p-hydroxyphenethylamine|3-Methoxy-4-hydroxyphenethylamine

Molecular weight: 203.7

CAS: 1477-68-5

Purity: ≥98%

Formulation: A crystalline solid

Product Type|Biochemicals|Receptor Pharmacology|Agonists||Research Area|Cancer||Research Area|Neuroscience|Neurodegenerative Disorders|Parkinson’s Disease||Research Area|Neuroscience|Neuroendocrinology

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