A phorboid vanilloid with capsaicin-like selectivity for the cloned rat TRPV1; induces Ca2+-uptake by rat dorsal root ganglion neurons (EC50 = 70 nM)

PDDHV – 5 mg

Brand:
Cayman
CAS:
179469-40-0
Storage:
4
UN-No:
- 2811 / 6.1

PDDHV is a resiniferatoxin-type phorboid vanilloid with capsaicin-like selectivity for the cloned rat transient receptor potential cation channel subfamily V member 1 (TRPV1), formerly known as vanilloid receptor 1.{32371} It induces Ca2+-uptake by rat dorsal root ganglion neurons with an EC50 value of 70 nM.{32371}  

 

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SKU: 20445 - Category:

Description

A phorboid vanilloid with capsaicin-like selectivity for the cloned rat TRPV1; induces Ca2+-uptake by rat dorsal root ganglion neurons (EC50 = 70 nM)

Formal name: 4-hydroxy-3-methoxy-[1aR,1bS,4aR,7aS,7bS,8R,9R,9aS-decahydro-4a,7b-dihydroxy-1,1,6,8-tetramethyl-5-oxo-9,9a-bis[(1-oxodecyl)oxy]-1H-cyclopropa[3,4]benz[1,2-e]azulen-3-yl]benzeneacetic acid,methyl ester

Synonyms:  Phorbol 12,13-didecanoate 20-homovanillate

Molecular weight: 837.1

CAS: 179469-40-0

Purity: ≥99%

Formulation: A solid

Product Type|Biochemicals|Ion Channel Modulation|Activators||Research Area|Neuroscience

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