A fluoroquinolone antibiotic that demonstrates extremely high potency against a wide range of bacteria in vitro; has an anionic structure

Delafloxacin – 25 mg

Brand:
Cayman
CAS:
189279-58-1
Storage:
-20
UN-No:
Non-Hazardous - /

Delafloxacin is a fluoroquinolone antibiotic that demonstrates extremely high potency against a wide range of bacteria in vitro, including levofloxacin-resistant strains of S. pneumoniae and methicillin-resistant S. aureus.{32844,32846} It targets both DNA gyrase and topoisomerase IV. Delafloxacin has an anionic structure, which enhances its potency in acidic environments (e.g., phagolysosome, inflammatory cells) and in skin and soft tissue infections.{32845}  

 

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Description

A fluoroquinolone antibiotic that demonstrates extremely high potency against a wide range of bacteria in vitro; has an anionic structure, which enhances its potency in acidic environments and in skin and soft tissue infections

Formal name: 1-(6-amino-3,5-difluoro-2-pyridinyl)-8-chloro-6-fluoro-1,4-dihydro-7-(3-hydroxy-1-azetidinyl)-4-oxo-3-quinolinecarboxylic acid

Synonyms:  ABT-492|RX-3341

Molecular weight: 440.8

CAS: 189279-58-1

Purity: 98%

Formulation: A crystalline solid

Product Type|Biochemicals|Antibiotics|Quinolones & Fluoroquinolones||Product Type|Biochemicals|Small Molecule Inhibitors|MMPs||Product Type|Biochemicals|Small Molecule Inhibitors|Nucleic Acid Turnover/Signaling||Research Area|Immunology & Inflammation||Research Area|Infectious Disease|Bacterial Diseases|MRSA

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