A potent inhibitor of PRMT4 (IC50 50 = 43 nM) in vitro

TP-064 – 25 mg

Brand:
Cayman
CAS:
2080306-20-1
Storage:
-20
UN-No:
Non-Hazardous - /

TP-064 is a potent inhibitor of protein arginine methyltransferase 4 (PRMT4; IC50 50 = 43 nM) in vitro. For more information on TP-064 please visit the Structural Genomics Consortium (SGC). The negative control, TP-064N, for TP-064 is also available exclusively through the SGC. You can submit a request to receive the negative control here.  

 

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SKU: 20256 - Category:

Description

A potent inhibitor of PRMT4 (IC50 50 = 43 nM) in vitro,

Formal name: N-methyl-N-[[2-[1-[2-(methylamino)ethyl]-4-piperidinyl]-4-pyridinyl]methyl]-3-phenoxy-benzamide

Synonyms: 

Molecular weight: 458.6

CAS: 2080306-20-1

Purity: ≥98%

Formulation: A crystalline solid

Product Type|Biochemicals|Small Molecule Inhibitors|Methyltransferases||Product Type|Biochemicals|Small Molecule Inhibitors|Nucleic Acid Turnover/Signaling||Research Area|Epigenetics, Transcription, & Translation|Writers|Histone Methylation

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