A glucose transporter inhibitor; selectively inhibits Glut4

BAY-588 – 1 mg

Brand:
Cayman
CAS:
1799759-24-2
Storage:
-20
UN-No:
Non-Hazardous - /

BAY-588 is a glucose transporter inhibitor and derivative of BAY-876 (Item No. 19961).{38214} It selectively inhibits glucose transporter 4 (Glut4), Glut1, and Glut3 over Glut2 with IC50 values of 0.5, 1.18, 5.47, and >10 μM, respectively, in CHO cells expressing human recombinant transporters.  

 

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SKU: 19960 - Category:

Description

A glucose transporter inhibitor; selectively inhibits Glut4, Glut1, and Glut3 over Glut2 (IC50s = 0.5, 1.18, 5.47, and >10 μM, respectively, in CHO cells expressing human recombinant transporters)

Formal name: N4-[1-[[4-(1,1-dimethylethyl)phenyl]methyl]-5-methyl-3-(trifluoromethyl)-1H-pyrazol-4-yl]-7-fluoro-2,4-quinolinedicarboxamide

Synonyms: 

Molecular weight: 527.5

CAS: 1799759-24-2

Purity: ≥98%

Formulation: A crystalline solid

Product Type|Biochemicals|Transporter & Exchanger Modulators||Research Area|Endocrinology & Metabolism|Carbohydrate Metabolism

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