Description
An inhibitor of Mps1 (IC50 = 145 nM); 1,000-fold selective for Mps1 over a panel of 352 kinases at 10 mM, but does inhibit Plk1 (Kd = 61 nM)
Formal name: 9-cyclopentyl-2-[[2-ethoxy-4-(4-hydroxy-1-piperidinyl)phenyl]amino]-5,7,8,9-tetrahydro-5-methyl-6H-pyrimido[4,5-b][1,4]diazepin-6-one
Synonyms:
Molecular weight: 480.6
CAS: 1228817-38-6
Purity: ≥98%
Formulation: A crystalline solid
Product Type|Biochemicals|Kinase Inhibitors|Other Serine/Threonine Kinases||Product Type|Biochemicals|Small Molecule Inhibitors|Kinases||Research Area|Cell Biology|Cell Cycle
