A stearoyl-CoA desaturase 1 inhibitor (IC50 = 6.3 nM) that induces cell death of hPSCs and inhibits the proliferation of human non-small cell lung carcinoma H1299 cells in vitro

A-939572 – 5 mg

Brand:
Cayman
CAS:
1032229-33-6
Storage:
-20
UN-No:
Non-Hazardous - /

A-939572 inhibits stearoyl-CoA desaturase 1 (IC50 = 6.3 nM), a key enzyme for lipid metabolism that is expressed in human pluripotent stem cells (hPSCs).{32308} This compound has been used to induce cell death of hPSCs as well as to inhibit the proliferation of human non-small cell lung carcinoma H1299 cells in vitro.{32308,26485}  

 

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Description

A stearoyl-CoA desaturase 1 inhibitor (IC50 = 6.3 nM) that induces cell death of hPSCs and inhibits the proliferation of human non-small cell lung carcinoma H1299 cells in vitro

Formal name: 4-(2-chlorophenoxy)-N-[3-[(methylamino)carbonyl]phenyl]-1-piperidinecarboxamide

Synonyms:  SCD1 Inhibitor|Stearoyl-CoA Desaturase 1 Inhibitor

Molecular weight: 387.9

CAS: 1032229-33-6

Purity: ≥98%

Formulation: A crystalline solid

Product Type|Biochemicals|Small Molecule Inhibitors|Fatty Acid Metabolism||Research Area|Cancer||Research Area|Cell Biology|Cell Death||Research Area|Cell Biology|Stem Cell Research||Research Area|Endocrinology & Metabolism

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