A methylated analog of SP 600125 that has much lower affinity for JNK isoforms (IC50s = 18 and 24 µM for JNK2 and JNK3

SP 600125, negative control – 1 mg

Brand:
Cayman
CAS:
54642-23-8
Storage:
-20
UN-No:
Non-Hazardous - /

SP 600125 (Item No. 10010466) is a selective, cell-permeable, reversible inhibitor of JNK isoforms 1-3 with Ki values of 0.19 μM.{16589} SP 600125, negative control is a methylated analog of SP 600125 that has much lower affinity for JNK isoforms (IC50s = 18 and 24 µM for JNK2 and JNK3, respectively).{16589}  

 

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Description

A methylated analog of SP 600125 that has much lower affinity for JNK isoforms (IC50s = 18 and 24 µM for JNK2 and JNK3, respectively)

Formal name: 2-methyl-dibenz[cd,g]indazol-6(2H)-one

Synonyms:  ​JNK Inhibitor II, negative control

Molecular weight: 234.3

CAS: 54642-23-8

Purity: ≥97%

Formulation: A solid

Product Type|Biochemicals|Kinase Inhibitors|Negative Controls||Product Type|Biochemicals|Small Molecule Inhibitors|Kinases||Research Area|Immunology & Inflammation|Adaptive Immunity||Research Area|Immunology & Inflammation|Innate Immunity

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