A proton pump inhibitor

Tenatoprazole – 50 mg

Brand:
Cayman
CAS:
113712-98-4
Storage:
-20
UN-No:
Non-Hazardous - /

Tenatoprazole is a proton pump inhibitor, blocking hog gastric H+/K+-ATPase activity with an IC50 value of 6.2 µM.{32337} It is orally bioavailable, blocking induced gastric acid secretion and ulcer formation in rats and humans.{32337,32335,32336} Tenatoprazole has a prolonged plasma half-life resulting in persistent effectiveness after withdrawal.{32336}  

 

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Description

A proton pump inhibitor, blocking hog gastric H+/K+-ATPase activity with an IC50 value of 6.2 µM; blocks induced gastric acid secretion and ulcer formation in rats and humans

Formal name: 5-methoxy-2-[[(4-methoxy-3,5-dimethyl-2-pyridinyl)methyl]sulfinyl]-3H-imidazo[4,5-b]pyridine

Synonyms:  TU-199

Molecular weight: 346.4

CAS: 113712-98-4

Purity: ≥98%

Formulation: A solid

Product Type|Biochemicals|Small Molecule Inhibitors|ATPases||Product Type|Biochemicals|Transporter & Exchanger Modulators

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