An agonist of the sigma-1 receptor (Ki = 10.4 nM); also binds the serotonin 5-HT3 and muscarinic acetylcholine receptors (Kis = 7.9 and 76 nM

Carbetapentane (citrate) – 100 mg

Brand:
Cayman
CAS:
23142-01-0
Storage:
-20
UN-No:
Non-Hazardous - /

Carbetapentane is an agonist of the sigma-1 receptor (Ki = 10.4 nM).{25816,21421} It also binds the serotonin 5-HT3 and muscarinic acetylcholine receptors (Kis = 7.9 and 76 nM, respectively).{30163,30164} Carbetapentane is a potent antitussive, anticonvulsant, and spasmolytic agent in clinical trials.{21421,30164}  

 

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Description

An agonist of the sigma-1 receptor (Ki = 10.4 nM); also binds the serotonin 5-HT3 and muscarinic acetylcholine receptors (Kis = 7.9 and 76 nM, respectively)

Formal name: 1-phenyl-cyclopentanecarboxylic acid 2-[2-(diethylamino)ethoxy]ethyl ester, 2-hydroxy-1,2,3-propanetricarboxylate

Synonyms:  Pentoxyverine citrate

Molecular weight: 525.6

CAS: 23142-01-0

Purity: ≥98%

Formulation: A crystalline solid

Product Type|Biochemicals|Ion Channel Modulation||Product Type|Biochemicals|Receptor Pharmacology||Product Type|Biochemicals|Small Molecule Activators||Research Area|Neuroscience|Seizure Disorders

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