A partial agonist at 5-HT1A

Eltoprazine (hydrochloride) – 5 mg

Brand:
Cayman
CAS:
98206-09-8
Storage:
-20
UN-No:
Non-Hazardous - /

Eltoprazine is a phenylpiperazine compound that acts as a partial agonist at serotonin 5-HT1A, 5-HT1B, and 5-HT2B receptors (Kis = 40, 52, and 81 nM, respectively).{29966} It exerts a dose-dependent decrease in aggressive behavior in resident-intruder tests with rats (ID50 = 0.24 mg/kg).{29965}  

 

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Description

A partial agonist at 5-HT1A, 5-HT1B, and 5-HT2B receptors (Kis = 40, 52, and 81 nM, respectively); decreases aggressive behavior in resident-intruder tests with rats (ID50 = 0.24 mg/kg)

Formal name: 1-(2,3-dihydro-1,4-benzodioxin-5-yl)-piperazine, monohydrochloride

Synonyms:  DU-28,853|DU-28,893

Molecular weight: 256.7

CAS: 98206-09-8

Purity: ≥98%

Formulation: A crystalline solid

Product Type|Biochemicals|Receptor Pharmacology|Agonists||Research Area|Neuroscience|Behavioral Neuroscience

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