A prodrug for terbutaline

Bambuterol (hydrochloride) – 1 g

Brand:
Cayman
CAS:
81732-46-9
Storage:
-20
UN-No:
Non-Hazardous - /

Bambuterol is a prodrug for terbutaline, a long-acting β-adrenoceptor agonist (Ki = 15.4 µM for human β2-adrenergic receptor).{25395} Bambuterol is converted to terbutaline by butyrylcholinesterases in the liver and plasma.{29051} Long-acting β agonists are useful in ameliorating symptoms of asthma.{29052}  

 

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Description

A prodrug for terbutaline, a long-acting β-adrenoceptor agonist (Ki = 15.4 µM for human β2-adrenergic receptor); converted to terbutaline by butyrylcholinesterases in the liver and plasma

Formal name: N,N-dimethyl-carbamic acid-3-[[(dimethylamino)carbonyl]oxy]-5-[2-[(1,1-dimethylethyl)amino]-1-hydroxyethyl]phenyl ester, monohydrochloride

Synonyms:  KWD 2183

Molecular weight: 403.9

CAS: 81732-46-9

Purity: ≥95%

Formulation: A crystalline solid

Product Type|Biochemicals|Receptor Pharmacology|Agonists||Research Area|Immunology & Inflammation|Pulmonary Diseases|Asthma

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