An agonist of dopamine D1A (D1R) and D1B (D5R) receptors (Kds = 17 and 11 nM

Fenoldopam (mesylate) – 5 mg

Brand:
Cayman
CAS:
67227-57-0
Storage:
-20
UN-No:
Non-Hazardous - /

Fenoldopam is an agonist of dopamine D1A (D1R) and D1B (D5R) receptors (Kds = 17 and 11 nM, respectively).{31154,31157} Fenoldopam is used to study the roles of these receptors, in cells and in vivo, and to alter hemodynamic properties, including hypertension, in animals.{31155,31156}  

 

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Description

An agonist of dopamine D1A (D1R) and D1B (D5R) receptors (Kds = 17 and 11 nM, respectively); alters hemodynamic properties, including hypertension, in animals.

Formal name: 6-chloro-2,3,4,5-tetrahydro-1-(4-hydroxyphenyl)-1H-3-benzazepine-7,8-diol, monomethanesulfonate

Synonyms:  SKF 82526J

Molecular weight: 401.9

CAS: 67227-57-0

Purity: ≥95%

Formulation: A crystalline solid

Product Type|Biochemicals|Receptor Pharmacology|Agonists||Research Area|Cardiovascular System|Cardiovascular Diseases|Hypertension||Research Area|Neuroscience

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