A synthetic CB structurally similar to UR-144

Azidoindolene 1 – 1 mg

Brand:
Cayman
CAS:
1364933-69-6
Storage:
-20
UN-No:
Non-Hazardous - /

UR-144 (Item No. 11502) and XLR11 (Item No. 11565) are potent synthetic cannabinoids (CBs) that have been identified as adulterants of herbal products.{22648,23290} Azidoindolene 1 is structurally similar to UR-144, XLR11, and a number of additional synthetic CBs with a hydrazide linking the tetramethylcyclopropyl group to the aminoalkylindole group. The physiological and toxicological properties of this compound are not known. Typically, a tetramethylcyclopropyl group confers selectivity for the peripheral CB2 receptor, and the addition of substituents at the N1-amine of the aminoalkylindole group is necessary for high affinity at either CB1 or CB2.{20487} This product is intended for forensic and research applications.  

 

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Description

A synthetic CB structurally similar to UR-144, XLR11, and a number of other synthetic CBs with a hydrazide linking the tetramethylcyclopropyl group to the aminoalkylindole group; intended for forensic and research applications

Formal name: 2,2,3,3-tetramethyl-cyclopropanecarboxylic acid (2Z)-2-[1-(5-fluoropentyl)-1,2-dihydro-2-oxo-3H-indol-3-ylidene]hydrazide

Synonyms: 

Molecular weight: 373.5

CAS: 1364933-69-6

Purity: ≥98%

Formulation: A crystalline solid

Application|Mass Spectrometry||Product Type|Biochemicals|Analytical Standards||Product Type|Biochemicals|Drugs of Abuse||Research Area|Forensic Chemistry & Toxicology|Cannabinoids|Synthetic Cannabinoids

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