11-keto Fluprostenol is an analog of PGD2 with structural modifications intended to give it a prolonged half-life and greater potency. Fluprostenol is a well-studied

11-keto Fluprostenol – 1 mg

Brand:
Cayman
CAS:
62145-07-7
Storage:
-20
UN-No:
De Minimis - 1231 / 3

11-keto Fluprostenol is an analog of prostaglandin D2 (PGD2) with structural modifications intended to give it a prolonged half-life and greater potency. Fluprostenol is a well-studied, potent analog of PGF2α and acts primarily through the FP receptor.{1182} Oxidation at C-11 of fluprostenol yields 11-keto fluprostenol. 11-keto Fluprostenol exhibits moderate binding to the CRTH2/DP2 receptor compared to PGD2 and essentially no activity at the DP1 receptor.{10723}  

 

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11-keto Fluprostenol is an analog of PGD2 with structural modifications intended to give it a prolonged half-life and greater potency. Fluprostenol is a well-studied, potent analog of PGF2α and acts primarily through the FP receptor.{1182} Oxidation at C-11 of fluprostenol yields 11-keto fluprostenol. 11-keto Fluprostenol exhibits moderate binding to the CRTH2/DP2 receptor compared to PGD2 and essentially no activity at the DP1 receptor.{10723}

Formal name: 11-oxo-9α,15R-dihydroxy-16-(3-(trifluoromethyl)phenoxy)-17,18,19,20-tetranor-prosta-5Z,13E-dien-1-oic acid

Synonyms:  Fluprostenol Prostaglandin D2

Molecular weight: 456.5

CAS: 62145-07-7

Purity: ≥98%

Formulation: A solution in methyl acetate

Product Type|Biochemicals|Lipids|Prostaglandins||Product Type|Biochemicals|Receptor Pharmacology||Research Area|Lipid Biochemistry|Cyclooxygenase Pathway

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