An antiviral prodrug targeted against the influenza viruses; once hydrolyzed to its active metabolite

Oseltamivir (phosphate) – 250 mg

Brand:
Cayman
CAS:
204255-11-8
Storage:
-20
UN-No:
Non-Hazardous - /

Oseltamivir is an antiviral prodrug targeted against the influenza viruses.{25827,25824} Once hydrolyzed in the liver to its active metabolite, oseltamivir acid (Item No. 15779), it can competitively inhibit viral neuraminidase (IC50s = 0.1-4.9 nM for influenza neuraminidases A and B), blocking the release of new viral particles from a host cell.{25825,25826,25830,25829,25828}  

 

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Description

An antiviral prodrug targeted against the influenza viruses; once hydrolyzed to its active metabolite, it can competitively inhibit viral neuraminidase (IC50s = 0.1-4.9 nM for influenza neuraminidases A and B)

Formal name: 4R-(acetylamino)-5S-amino-3R-(1-ethylpropoxy)-1-cyclohexene-1-carboxylic acid, ethyl ester, monophosphate

Synonyms:  GS-4104|Ro 64-0796/002|Tamiflu®

Molecular weight: 410.4

CAS: 204255-11-8

Purity: ≥98%

Formulation: A crystalline solid

Product Type|Biochemicals|Antivirals|Neuraminidase Inhibitors||Product Type|Biochemicals|Small Molecule Inhibitors||Research Area|Immunology & Inflammation||Research Area|Infectious Disease|Viral Diseases|Influenza

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