The active metabolite of the antiviral prodrug oseltamivir; acts as an inhibitor of influenza neuraminidases A and B (IC50 values are 0.1 to 4.9 nM for both enzymes)

Oseltamivir Acid – 5 mg

Brand:
Cayman
CAS:
187227-45-8
Storage:
-20
UN-No:
Non-Hazardous - /

Oseltamivir (GS-4104) is an antiviral prodrug targeted against the influenza viruses.{25827,25824} Oseltamivir acid is the active metabolite of oseltamivir.{25825,25826} It acts as an inhibitor of influenza neuraminidases A and B (IC50 = 0.1 to 4.9 nM for both enzymes), in this way preventing virus budding and release.{25830,25829,25828}  

 

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Description

The active metabolite of the antiviral prodrug oseltamivir; acts as an inhibitor of influenza neuraminidases A and B (IC50 values are 0.1 to 4.9 nM for both enzymes), in this way preventing virus budding and release

Formal name: 4R-(acetylamino)-5S-amino-3R-(1-ethylpropoxy)-1-cyclohexene-1-carboxylic acid

Synonyms:  GS-4071|Ro 64-0802

Molecular weight: 284.4

CAS: 187227-45-8

Purity: ≥95%

Formulation: A crystalline solid

Product Type|Biochemicals|Antivirals|Neuraminidase Inhibitors||Product Type|Biochemicals|Small Molecule Inhibitors||Research Area|Immunology & Inflammation||Research Area|Infectious Disease|Viral Diseases|Influenza

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