The racemic mixture of the water soluble

(±)-ORG 28611 – 5 mg

Brand:
Cayman
CAS:
784138-08-5
Storage:
-20
UN-No:
Non-Hazardous - /

(±)-ORG 28611 is the racemic mixture of the water soluble, full agonist of the human cannabinoid (CB) receptors central CB1 (pEC50 = 7.6; pKi = 8.9) and peripheral CB2 (pKi = 8.8).{23926} ORG 28611 (0.1-1 μM/kg, intravenous) demonstrated antinociceptive activity in the mouse tail flick test and the mouse formalin paw test, and it was further evaluated clinically for use as a potential intravenous analgesic agent.{23926}  

 

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Description

The racemic mixture of the water soluble, full agonist of the human CB receptors central CB1 (pEC50 = 7.6; pKi = 8.9) and peripheral CB2 (pKi = 8.8); demonstrates antinociceptive activity in the mouse tail flick test and the mouse formalin paw test

Formal name: [1-(cyclohexylmethyl)-7-methoxy-1H-indol-3-yl](3,4-dimethyl-1-piperazinyl)-methanone

Synonyms: 

Molecular weight: 383.5

CAS: 784138-08-5

Purity: ≥98%

Formulation: A crystalline solid

Application|Mass Spectrometry||Product Type|Biochemicals|Analytical Standards||Product Type|Biochemicals|Drugs of Abuse||Research Area|Forensic Chemistry & Toxicology|Cannabinoids|Synthetic Cannabinoids

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