A potent inhibitor of chymotrypsin and chymase (Ki = 9.36 and 13.1 nM

Chymostatin – 5 mg

Brand:
Cayman
CAS:
9076-44-2
Storage:
-20
UN-No:
Non-Hazardous - /

Chymostatin is a bioactive peptide of microbial origin that acts as a protease inhibitor with selectivity for chymotryptase-like serine proteases.{24067} It potently inhibits chymotrypsin and chymase (Ki = 9.36 and 13.1 nM, respectively) while less effectively blocking the activity of cathepsins, papain, and leukocyte elastase.{24069,24067,24065,24068,24066} It is without effect on trypsin, thrombin, plasmin, pepsin, and kallikrein.{24067}  

 

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Description

A potent inhibitor of chymotrypsin and chymase (Ki = 9.36 and 13.1 nM, respectively), that less effectively blocks the activity of cathepsins, papain, and leukocyte elastase

Formal name:

Synonyms: 

Molecular weight: 607.7

CAS: 9076-44-2

Purity: ≥95% (a mixture of A, B, C)

Formulation: A crystalline solid

Product Type|Biochemicals|Peptides||Product Type|Biochemicals|Small Molecule Inhibitors|MMPs||Product Type|Biochemicals|Small Molecule Inhibitors|Peptidases & Proteases||Research Area|Cell Biology|Proteolysis

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