An agonist of both nAChR and mAChR receptors

Carbamoylcholine (chloride) – 1 g

Brand:
Cayman
CAS:
51-83-2
Storage:
-20
UN-No:
De Minimis - 2811 / 6.1

Carbamoylcholine, also known as carbachol, is an analog of acetylcholine that activates acetylcholine receptors (AChR). Carbamoylcholine is an agonist of both nicotinic (nAChR) and muscarinic (mAChR) receptors, with reported Ki values ranging from 10 to 10,000 nM for different receptors and different preparations.{27179,27173,27178,27174,27175} Carbamoylcholine (chloride) is used to study responses mediated by nAChR and mAChR, including smooth muscle contraction, gut motility, and neuronal signaling.{27180,27177,27176}  

 

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Description

An agonist of both nAChR and mAChR receptors, with reported Ki values ranging from 10 to 10,000 nM for different receptors and different preparations; used to study responses mediated by nAChR and mAChR, including smooth muscle contraction, gut motility, and neuronal signaling

Formal name: 2-[(aminocarbonyl)oxy]-N,N,N-trimethyl-ethanaminium, monochloride

Synonyms:  Carbachol

Molecular weight: 182.7

CAS: 51-83-2

Purity: ≥98%

Formulation: A crystalline solid

Product Type|Biochemicals|Ion Channel Modulation|Activators||Product Type|Biochemicals|Receptor Pharmacology|Agonists||Research Area|Neuroscience

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