A 2C-I derivative that acts as a partial agonist of human 5-HT2A receptors (Ki = 0.26 nM; EC50 = 1.6 nM); intended for forensic and research applications

25I-NBF (hydrochloride) – 5 mg

Brand:
Cayman
CAS:
1539266-13-1
Storage:
-20
UN-No:
Non-Hazardous - /

25I-NBF is an N-benzyl derivative of the phenethylamine hallucinogen 2C-I which acts as a highly potent partial agonist for the 5-HT2A receptor. 25I-NBF acts as a partial agonist of human 5-HT2A receptors demonstrating a Ki value of 0.26 nM and an EC50 value of 1.6 nM.{20442} A radiolabelled form of 25I-NBF has been used for mapping the distribution of 5-HT2A receptors in the brain, using positron emission tomography.{21331} This product is intended for forensic and research applications.  

 

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Description

A 2C-I derivative that acts as a partial agonist of human 5-HT2A receptors (Ki = 0.26 nM; EC50 = 1.6 nM); intended for forensic and research applications

Formal name: N-(2-fluorobenzyl)-2-(4-iodo-2,5-dimethoxyphenyl)ethanamine, monohydrochloride

Synonyms:  2C-I-NBF

Molecular weight: 451.7

CAS: 1539266-13-1

Purity: ≥98%

Formulation: A crystalline solid

Application|Mass Spectrometry||Product Type|Biochemicals|Analytical Standards||Product Type|Biochemicals|Drugs of Abuse||Research Area|Forensic Chemistry & Toxicology|Hallucinogens|Phenethylamines||Research Area|Forensic Chemistry & Toxicology|Stimulants|Phenethylamines

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