An ACE inhibitor (IC50 = 0.93 nM)

Trandolapril – 250 mg

Brand:
Cayman
CAS:
87679-37-6
Storage:
-20
UN-No:
Non-Hazardous - /

Trandolapril is an inhibitor of angiotensin-converting enzyme (ACE; IC50 = 0.93 nM).{23056} Formulations containing trandolapril, with or without the calcium channel blocker verapamil (Item No. 14288), are effective against certain cardiovascular disorders, including essential hypertension.{33810,33812} ACE inhibitors, including trandolapril, also have neuroprotective effects in animal models.{33811}  

 

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Description

An ACE inhibitor (IC50 = 0.93 nM)

Formal name: (2S,3aR,7aS)-1-[(2S)-2-[[(1S)-1-(ethoxycarbonyl)-3-phenylpropyl]amino]-1-oxopropyl]octahydro-1H-indole-2-carboxylic acid

Synonyms:  RU-44570

Molecular weight: 430.5

CAS: 87679-37-6

Purity: ≥98%

Formulation: A crystalline solid

Product Type|Biochemicals|Small Molecule Inhibitors|Angiotensin-converting Enzyme||Product Type|Biochemicals|Small Molecule Inhibitors|MMPs||Research Area|Cardiovascular System|Cardiovascular Diseases|Hypertension||Research Area|Neuroscience|Neuroprotection

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