A bicyclic CB analog with potent analgesic activity; comparable or more potent than Δ9-THC in analgesic

(-)-CP 47,497 (exempt preparation) – 10 mg

Brand:
Cayman
CAS:
114753-51-4
Storage:
-20
UN-No:
De Minimis - 1230 / 3|6.1

CP 47,497 is a bicyclic cannabinoid analog with potent analgesic activity.{16402} It is comparable or more potent than Δ9-tetrahydrocannabinol in analgesic, motor depressant, anticonvulsant and hypothermic effects in mice, rats, and dogs.{17029} The levorotatory enantiomer, (−)-CP 47,497 avidly binds the CB1 receptor (Ki = 2.1 nM).{17030}  

 

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Description

A bicyclic CB analog with potent analgesic activity; comparable or more potent than Δ9-THC in analgesic, motor depressant, anticonvulsant, and hypothermic effects; avidly binds the central cannabinoid receptor CB1 receptor (Ki = 2.1 nM).

Formal name: 2[(1S,3R)-3-hydroxycyclohexyl]-5-(2-methyloctan-2-yl)phenol

Synonyms: 

Molecular weight: 318.5

CAS: 114753-51-4

Purity: ≥98%

Formulation: A solution in methanol

Product Type|Biochemicals|Drugs of Abuse||Research Area|Forensic Chemistry & Toxicology|Cannabinoids|Synthetic Cannabinoids

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