An antimalarial compound and derivative of artemisinin; inhibits P. falciparum (IC50 = 1.27 nM in vitro); effective against various strains of P. berghei in mice (ED90 = 0.5-8.2 nM)

Arteether – 5 mg

Brand:
Cayman
CAS:
75887-54-6
Storage:
-20
UN-No:
Non-Hazardous - /

Arteether is a derivative of the antimalarial drug artemisinin (Item No. 11816). Arteether inhibits P. falciparum with an IC50 value of 1.27 nM in vitro.{39374} It is effective against various strains of P. berghei in mice with ED90 values of 0.5-8.2 nM.  

 

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SKU: 11814 - 5 mg Category:

Description

An antimalarial compound and derivative of artemisinin; inhibits P. falciparum (IC50 = 1.27 nM in vitro); effective against various strains of P. berghei in mice (ED90 = 0.5-8.2 nM) ,

Formal name: (3R,5aS,6R,8aS,9R,10S,12R,12aR)-10-ethoxydecahydro-3,6,9-trimethyl-3,12-epoxy-12H-pyrano[4,3-j]-1,2-benzodioxepin

Synonyms:  Artemotil|Dihydroartemisinin ethyl ether|NSC 665971

Molecular weight: 312.4

CAS: 75887-54-6

Purity: ≥95%

Formulation: A crystalline solid

Product Type|Biochemicals|Antiparasitics|Antiprotozoals||Research Area|Immunology & Inflammation||Research Area|Infectious Disease|Parasitic Diseases|Malaria

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