A dual 5-LO and mPGES-1 inhibitor (IC50s = 1 and 3.6 µM

1-Naphthyl 3,5-dinitrobenzoate – 10 mg

Brand:
Cayman
CAS:
93261-39-3
Storage:
-20
UN-No:
Non-Hazardous - /

1-Naphthyl 3,5-dinitrobenzoate has been identified as a dual 5-lipoxygenase and microsomal prostaglandin E synthase-1 inhibitor with IC50 values of 1 and 3.6 µM, respectively.{20842} The scaffold of this compound is being explored for anti-inflammatory drug design.{20842}  

 

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SKU: 11729 - 10 mg Category:

Description

A dual 5-LO and mPGES-1 inhibitor (IC50s = 1 and 3.6 µM, respectively),

Formal name: 1-(3,5-dinitrobenzoate) 1-naphthalenol

Synonyms:  1-(3,5-Dinitrobenzoyloxy)naphthalene|1-Naphthalonol 3,5-dinitrobenzoate

Molecular weight: 338.3

CAS: 93261-39-3

Purity: ≥98%

Formulation: A crystalline solid

Product Type|Biochemicals|Small Molecule Inhibitors|Lipoxygenases||Product Type|Biochemicals|Small Molecule Inhibitors|Prostaglandin Synthases||Research Area|Immunology & Inflammation|Inflammatory Lipid Mediators|Prostaglandins||Research Area|Lipid Biochemistry|Cyclooxygenase Pathway||Research Area|Lipid Biochemistry|Lipoxygenase Pathways

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