A diterpene with diverse biological activities; activates rat adipocyte adenylyl cyclase (IC50 = 20 µM); inhibits glucose transport in rat adipocyte plasma membranes; reduces blood pressure in spontaneously hypertensive rats from 30-1

Deacetylforskolin – 5 mg

Brand:
Cayman
CAS:
64657-20-1
Storage:
-20
UN-No:
Non-Hazardous - /

Deacetylforskolin is a diterpene and a derivative of forskolin (Item No. 11018) that has been found in C. forskohlii and has diverse biological activities.{52583,34031,41421,52584} It activates rat adipocyte adenylyl cyclase (IC50 = 20 µM) and inhibits glucose transport in rat adipocyte plasma membranes.{34031} Deactylforskolin (30-1,000 µg/kg) reduces blood pressure in spontaneously hypertensive rats.{41421} It also attenuates hypercapnia-induced impairments in the passive avoidance response in mice.{52584}  

 

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SKU: 11701 - 5 mg Category:

Description

A diterpene with diverse biological activities; activates rat adipocyte adenylyl cyclase (IC50 = 20 µM); inhibits glucose transport in rat adipocyte plasma membranes; reduces blood pressure in spontaneously hypertensive rats from 30-1,000 µg/kg; attenuates hypercapnia-induced impairments in the passive avoidance response in mice

Formal name: (3R,4aR,5S,6S,6aS,10S,10aR,10bS)-3-ethenyldodecahydro-5,6,10,10b-tetrahydroxy-3,4a,7,7,10a-pentamethyl-1H-naphtho[2,1-b]pyran-1-one

Synonyms:  7-Deactylcoleonol|Forskolin D

Molecular weight: 368.5

CAS: 64657-20-1

Purity: ≥98%

Formulation: A solid

Product Type|Biochemicals|Natural Products|Terpenes||Product Type|Biochemicals|Small Molecule Activators|Cyclases||Research Area|Cardiovascular System|Cardiovascular Diseases|Hypertension||Research Area|Endocrinology & Metabolism||Research Area|Neuroscience|Behavioral Neuroscience|Learning & Memory

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