A potent psychoactive analog of 5-methoxy DiPT and AMT that inhibits re-uptake (IC50s = 0.18

5-methoxy AMT – 5 mg

Brand:
Cayman
CAS:
1137-04-8
Storage:
-20
UN-No:
Non-Hazardous - /

5-methoxy AMT (5-MeO AMT) is a potent psychoactive analog of 5-methoxy DiPT (Item No. 11865) and α-methyltryptamine (AMT), tryptamine derivatives that inhibit reuptake and stimulate release of monoamines.{19758} 5-MeO AMT inhibits re-uptake (IC50s = 0.18, 2.9, and 3.37 μM) and stimulates release (EC50s = 1.5, 460, and 8.9 μM) of dopamine, serotonin, and norepinephrine, respectively from rat brain synaptosomes.{19758} 5-MeO AMT, sometimes called Alpha-O, has been sold under the guise of LSD and abused as a recreational drug.{21059} This tryptamine analog is intended only to be used to aid the forensic analysis of samples that may contain this compound or for scientific research applications.  

 

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Description

A potent psychoactive analog of 5-methoxy DiPT and AMT that inhibits re-uptake (IC50s = 0.18, 2.9, and 3.37 μM) and stimulates release (EC50s = 1.5, 460, and 8.9 μM) of dopamine, serotonin, and norepinephrine, respectively from rat brain synaptosomes

Formal name: 5-methoxy-α-methyl-1H-indole-3-ethanamine

Synonyms:  5-MeO AMT

Molecular weight: 204.3

CAS: 1137-04-8

Purity: ≥98%

Formulation: A crystalline solid

Product Type|Biochemicals|Drugs of Abuse||Research Area|Forensic Chemistry & Toxicology|Hallucinogens|Tryptamines

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