A cannabimimetic indole with 5-fold selectivity for the CB1 receptor (Ki = 17 nM) compared to the CB2 receptor (Ki = 89 nM); stimulates GTPγS binding of CB1 and CB2 receptors with EC50 values of 29.3 and 24.4 nM

JWH 302 – 5 mg

Brand:
Cayman
CAS:
864445-45-4
Storage:
-20
UN-No:
De Minimis - 1231 / 3

JWH 302 is a cannabimimetic indole that shows 5-fold selectivity for the central cannabinoid (CB1) receptor with a Ki value of 17 nM compared to the peripheral cannabinoid (CB2) receptor (Ki = 89 nM).{17655} JWH 302 stimulates GTPγS binding of CB1 and CB2 receptors with EC50 values of 29.3 and 24.4 nM, respectively.{17655}  

 

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SKU: 10722 - 5 mg Category:

Description

A cannabimimetic indole with 5-fold selectivity for the CB1 receptor (Ki = 17 nM) compared to the CB2 receptor (Ki = 89 nM); stimulates GTPγS binding of CB1 and CB2 receptors with EC50 values of 29.3 and 24.4 nM, respectively

Formal name: 2-(3-methoxyphenyl)-1-(1-pentyl-1H-indol-3-yl)-ethanone

Synonyms: 

Molecular weight: 335.4

CAS: 864445-45-4

Purity: ≥95%

Formulation: A solution in methyl acetate

Product Type|Biochemicals|Drugs of Abuse||Research Area|Forensic Chemistry & Toxicology|Cannabinoids|Synthetic Cannabinoids

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