A potent CB receptor agonist that avidly binds to both CB1 and CB2 (Ki = 9.5 and 2.9 nM

JWH 007 – 5 mg

Brand:
Cayman
CAS:
155471-10-6
Storage:
-20
UN-No:
De Minimis - 1230 / 3|6.1

JWH 007 is a potent cannabinoid (CB) receptor agonist that avidly binds to both CB1 and CB2 (Ki = 9.5 and 2.9 nM, respectively).{18231,18232} This compares favorably with the binding of Δ9-THC, which binds CB1 and CB2 with Ki values of 41 and 36 nM, respectively.{18232} Similarly, JWH 007 performs comparably to Δ9-THC in mouse studies on spontaneous activity, antinociception, hypothermia, and catalepsy.{18231}  

 

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SKU: 10266 - 5 mg Category:

Description

A potent CB receptor agonist that avidly binds to both CB1 and CB2 (Ki = 9.5 and 2.9 nM, respectively); performs comparably to Δ9-THC in mouse studies on spontaneous activity, antinociception, hypothermia, and catalepsy

Formal name: (2-methyl-1-pentyl-1H-indol-3-yl)-1-naphthalenyl-methanone

Synonyms: 

Molecular weight: 355.5

CAS: 155471-10-6

Purity: ≥98%

Formulation: A solution in methanol

Application|Mass Spectrometry||Product Type|Biochemicals|Analytical Standards||Product Type|Biochemicals|Drugs of Abuse||Research Area|Forensic Chemistry & Toxicology|Cannabinoids|Synthetic Cannabinoids

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