An analog of bimatoprost

17-phenyl trinor Prostaglandin F2α methyl amide – 1 mg

Brand:
Cayman
CAS:
155206-01-2
Storage:
-20
UN-No:
De Minimis - 1170 / 3

17-phenyl trinor Prostaglandin F2α (17-phenyl trinor PGF2α) is a metabolically stable analog of PGF2α and is a potent agonist for the FP receptor, binding with a relative potency of 756% compared to that of PGF2α.{2058} The ethyl amide of 17-phenyl trinor PGF2α bimatoprost has been approved for use as an ocular hypotensive drug.{8941} 17-phenyl trinor PGF2α methyl amide is an analog of bimatoprost. Its biological and toxicological properties have not been evaluated.  

 

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SKU: 10010351 - 1 mg Category:

Description

An analog of bimatoprost

Formal name: (5Z)-7-[(1R,2R,3R,5S)-3,5-dihydroxy-2-[(1E,3S)-3-hydroxy-5-phenyl-1-penten-1-yl]cyclopentyl]-N-methyl-5-heptenamide

Synonyms:  17-phenyl trinor PGF2α methyl amide|Bimatoprost methyl amide|Methylamido Dihydro Noralfaprostal

Molecular weight: 401.5

CAS: 155206-01-2

Purity: ≥98%

Formulation: A solution in ethanol

Product Type|Biochemicals|Lipids|Prostaglandins||Research Area|Lipid Biochemistry|Cyclooxygenase Pathway||Research Area|Neuroscience|Ophthalmology

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