A stable analog of Δ9-THC and AEA; exhibits high-affinity for the CB1 and CB2 receptors (Ki = 210 and 30 nM

CB-52 – 1 mg

Brand:
Cayman
CAS:
869376-90-9
Storage:
-20
UN-No:
Non-Hazardous - /

CB-52 is a stable analog of Δ9-tetrahydrocannabinol (THC) and anandamide (AEA). It exhibits high affinity for the central cannabinoid (CB1) and peripheral cannabinoid (CB2) receptors with Ki values of 210 and 30 nM, respectively.{14815} In vitro, CB-52 behaves primarily as a CB1 receptor partial agonist and a CB2 receptor neutral antagonist.{14816}  

 

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SKU: 10010117 - 1 mg Category:

Description

A stable analog of Δ9-THC and AEA; exhibits high-affinity for the CB1 and CB2 receptors (Ki = 210 and 30 nM, respectively); behaves primarily as a CB1 receptor partial agonist and a CB2 receptor neutral antagonist in vitro

Formal name: N-cyclopropyl-11-(2-hexyl-5-hydroxyphenoxy)-undecanamide

Synonyms: 

Molecular weight: 417.6

CAS: 869376-90-9

Purity: ≥98%

Formulation: A crystalline solid

Application||Product Type|Biochemicals|Receptor Pharmacology|Agonists||Product Type|Biochemicals|Receptor Pharmacology|Antagonists||Research Area|Neuroscience|Cannabinoid Research|CB1 & CB2 Receptors

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