A lipophilic analog of 17-trifluoromethylphenyl trinor PGF2α

17-trifluoromethylphenyl trinor Prostaglandin F2α ethyl amide – 50 mg

Brand:
Cayman
CAS:
1621369-73-0
Storage:
-20
UN-No:
De Minimis - 1170 / 3

Prostaglandin F2α (PGF2α), acting through the FP receptor, causes smooth muscle contraction and exhibits potent luteolytic activity.{187,421,1651} 17-trifluoromethylphenyl trinor Prostaglandin F2α (17-trifluoromethylphenyl trinor PGF2α) is an analog of PGF2α that shares the meta-trifluoromethyl group of travoprost with the 17-phenyl trinor modification of latanoprost. It is anticipated to be a potent and selective agonist of the FP receptor, with potential applications in glaucoma and luteolysis. 17-trifluoromethylphenyl trinor PGF2α ethyl amide is a lipophilic analog of 17-trifluoromethylphenyl trinor PGF2α. Ethyl amides of PGs can serve as prodrugs, as they are hydrolyzed in certain tissues to generate the bioactive free acid.  

 

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SKU: 10010061 - 50 mg Category:

Description

A lipophilic analog of 17-trifluoromethylphenyl trinor PGF2α

Formal name: 9α,11α,15S-trihydroxy-17-trifluoromethylphenyl-18,19,20-trinor-prosta-5Z,13E-dien-1-oic acid, ethyl amide

Synonyms:  17-trifluoromethylphenyl trinor PGF2α ethyl amide

Molecular weight: 483.6

CAS: 1621369-73-0

Purity: >98%

Formulation: A solution in ethanol

Product Type|Biochemicals|Lipids|Prostaglandins||Research Area|Endocrinology & Metabolism|Reproductive Biology||Research Area|Lipid Biochemistry|Cyclooxygenase Pathway||Research Area|Neuroscience|Ophthalmology

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