Derivative of PGF1α containing a thio-fluorobenzene substituent in the lower side chain; binds to the recombinant human FP receptor with an IC50 value of about 30 nM

CAY10509 – 500 µg

Brand:
Cayman
CAS:
1245699-47-1
Storage:
-20
UN-No:
De Minimis - 1173 / 3

The actions of many clinical prostaglandins, including those used for estrous synchronization and for reduction of intraocular pressure, are mediated through the FP receptor.{2959} CAY10509 is an analog of PGF2α containing a thio-fluorobenzene substituent in the lower side chain. CAY10509 has an IC50 of about 30 nM when tested for binding to the recombinant human FP receptor.{14404}  

 

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SKU: 10009167 - 500 µg Category:

Description

Derivative of PGF1α containing a thio-fluorobenzene substituent in the lower side chain; binds to the recombinant human FP receptor with an IC50 value of about 30 nM

Formal name: 9α,11α,15R-trihydroxy-17-thiofluorophenoxy-17,18,19,20-tetranor-prostan-1-oic acid, methyl ester

Synonyms: 

Molecular weight: 442.6

CAS: 1245699-47-1

Purity: ≥98%

Formulation: A solution in ethyl acetate

Product Type|Biochemicals|Lipids|Prostaglandins||Product Type|Biochemicals|Receptor Pharmacology|Agonists||Research Area|Lipid Biochemistry|Cyclooxygenase Pathway

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