A potent

LY2183240 – 5 mg

Brand:
Cayman
CAS:
874902-19-9
Storage:
-20
UN-No:
Non-Hazardous - /

LY2183240 is a potent, competitive inhibitor of anandamide uptake (IC50 = 270 pM; Ki = 540 pM) and hydrolysis.{14134,15431,16339} It increases anandamide levels in rat cerebellum (ED50 = 1.37 mg/kg) and displays dose-dependent efficacy (3-30 mg/kg) in several rodent models of persistent pain.{14134}  

 

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SKU: 10008663 - 5 mg Category:

Description

A potent, competitive inhibitor of anandamide uptake (IC50 = 270 pM; Ki = 540 pM) and hydrolysis; increases anandamide levels in rat cerebellum (ED50 = 1.37 mg/kg) and displays dose-dependent efficacy (3-30 mg/kg) in several rodent models of persistent pain

Formal name: 5-([1,1′-biphenyl]-4-ylmethyl)-N,N-dimethyl-1H-tetrazole-1-carboxamide

Synonyms: 

Molecular weight: 307.4

CAS: 874902-19-9

Purity: ≥98%

Formulation: A crystalline solid

Application||Product Type|Biochemicals|Transporter & Exchanger Modulators||Research Area|Neuroscience|Cannabinoid Research|Endocannabinoids||Research Area|Neuroscience|Pain Research

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