3-HPA is an analog of AM404

N-(3-hydroxyphenyl)-Arachidonoyl amide – 100 mg

Brand:
Cayman
CAS:
183718-75-4
Storage:
-20
UN-No:
Excepted Quantity - 1170 / 3

N-(3-hydroxyphenyl)-Arachidonoyl amide (3-HPA) is an analog of AM404 (N-(4-hydroxyphenyl)-arachidonoyl amide), which is a selective inhibitor of carrier-mediated transport of arachidonoyl ethanolamide (AEA).{4894} 3-HPA is metabolized by both cyclooxygenase-1 (COX-1) and COX-2 and was found to selectively and irreversibly inhibit COX-2 with an IC50 value of 2 µM.{14589}  

 

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SKU: 10007704 - 100 mg Category:

Description

3-HPA is an analog of AM404, which is a selective inhibitor of carrier-mediated transport of AEA. 3-HPA is metabolized by both COX-1 and COX-2 and also selectively and irreversibly inhibits COX-2 with an IC50 value of 2 µM.

Formal name: N-(3-hydroxyphenyl)-5Z,8Z,11Z,14Z-eicosatetraenamide

Synonyms:  3-HPAA

Molecular weight: 395.6

CAS: 183718-75-4

Purity: >98%

Formulation: A solution in ethanol

Product Type|Biochemicals|Lipids|Fatty Amides||Product Type|Biochemicals|Small Molecule Inhibitors|Cyclooxygenases||Research Area|Lipid Biochemistry|Cyclooxygenase Pathway||Research Area|Neuroscience|Cannabinoid Research|Endocannabinoids

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