A synthetic CB that is selective for the peripheral CB2 receptor (Ki = 3.4 nM) over the central CB1 receptor (Ki = 677 nM); inhibits the growth of tumors in mice

JWH 133 – 10 mg

Brand:
Cayman
CAS:
259869-55-1
Storage:
-20
UN-No:
De Minimis - 1231 / 3

JWH 133 is a synthetic cannabinoid (CB) that is over 200-fold selective for the peripheral CB2 receptor (Ki = 3.4 nM) over the central CB1 receptor (Ki = 677 nM).{19286} It inhibits the growth of tumors in mice, increasing apoptosis and impairing angiogenesis.{10777,13625} JWH 133 also suppresses inflammation in experimental colitis and pancreatitis in mice as well as in in vitro models.{24680,24678,24679}  

 

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SKU: 10005428 - 10 mg Category:

Description

A synthetic CB that is selective for the peripheral CB2 receptor (Ki = 3.4 nM) over the central CB1 receptor (Ki = 677 nM); inhibits the growth of tumors in mice, increasing apoptosis and impairing angiogenesis; suppresses inflammation in experimental colitis and pancreatitis in mice

Formal name: 3-(1,1-dimethylbutyl)-6aR,7,10,10aR-tetrahydro-6,6,9-trimethyl-6H-dibenzo[b,d]pyran

Synonyms: 

Molecular weight: 312.5

CAS: 259869-55-1

Purity: ≥95%

Formulation: A solution in methyl acetate

Application|Mass Spectrometry||Product Type|Biochemicals|Analytical Standards||Product Type|Biochemicals|Drugs of Abuse||Research Area|Cancer|Angiogenesis||Research Area|Cancer|Cell Death|Apoptosis||Research Area|Forensic Chemistry & Toxicology|Cannabinoids|Synthetic Cannabinoids

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